Barasertib (AZD1152-HQPA)

Barasertib (AZD1152-HQPA)

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Barasertib (AZD1152-HQPA) is a highly selective Aurora B inhibitor with IC50 of 0.37 nM in a cell-free assay, ~3700 fold more selective for Aurora B over Aurora A. Phase 1.

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