Bromosporine
Bromosporine is a broad spectrum inhibitor for bromodomains with IC50 of 0.41 ?M, 0.29 ?M, 0.122 ?M and 0.017 ?M for BRD2, BRD4, BRD9 and CECR2, respectively.
Bromosporine is a broad spectrum inhibitor for bromodomains with IC50 of 0.41 ?M, 0.29 ?M, 0.122 ?M and 0.017 ?M for BRD2, BRD4, BRD9 and CECR2, respectively.