Tofacitinib (CP-690550) Citrate

Tofacitinib (CP-690550) Citrate

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Tofacitinib citrate (CP-690550 citrate) is a novel inhibitor of JAK with IC50 of 1 nM, 20 nM and 112 nM against JAK3, JAK2, and JAK1, respectively.

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